Selank

Also known as · TP-7 · tuftsin-derived heptapeptide anxiolytic (Institute of Molecular Genetics, Russia)

01 / Dosing schedule

Cited dosing

Selank has published human anxiety trial data from Russian groups, including a randomized comparison against medazepam, but no Western regulatory review. The dose reported in a European Psychiatry congress abstract is 2700 microg/day intranasally, with 900 microg as a single dose.

Selank in generalized anxiety disorder — intranasal

PhaseDose & frequency
Daily dose2700 microg/day intranasally
Single dose used for EEG assessment900 microg
Time to rapid responsedays 1-3 in 40% of patients (rapid responders)
Time to response in conventional respondersday 14
Total treatment durationn.a. — not stated in the abstract
Comparator trial (Zozulia 2008)selank (n=30) vs medazepam (n=32) in 62 patients with GAD and neurasthenia; Selank dose n.a. in that abstract

Source · Syunyakov T, Teleshova ES, Neznamov GG, Bochkarev VK. P-1114 — Rapid and Slow Response During Treatment of Generalized Anxiety Disorder With Peptide Anxiolytic Selank. European Psychiatry. 2012;27(S1). ↗

Source indication · Generalized anxiety disorder (and neurasthenia) — Russian clinical trials

Injection frequency
Daily intranasal dosing; the 2700 microg/day figure is a daily total, and the split across instillations is not stated in the abstract.
Injection sites
Not an injection in the cited trials: Selank was administered intranasally. No anatomical injection site exists in the source material.

02 / Reconstitution

Reconstitution reference

The Russian trials used a prepared intranasal Selank solution; no reconstitution procedure is published in either cited source.

Vialn.a. — trials used prepared intranasal solution
BAC watern.a.
Concentrationn.a.
Example dose2700 microg/day (trial daily dose)
On a U‑100 syringemicrog/day, intranasal
Open the reconstitution calculator →

03 / Overview

Protocol overview

Selank is a synthetic heptapeptide built from the immunomodulatory tetrapeptide tuftsin with a Pro-Gly-Pro stabilising tail. It is described in the European Psychiatry abstract as approved (in Russia) for the treatment of generalized anxiety disorder; it has no FDA or EMA approval.

The dose that can actually be cited is 2700 microg/day intranasally, in a study of 20 patients aged 24-52 with DSM-IV generalized anxiety disorder. A single 900 microg dose was used for the EEG substudy. Forty percent of patients were classed as rapid responders within days 1-3; the remaining 60% reached clinically significant change by day 14.

The best-known controlled trial, Zozulia and colleagues in Zh Nevrol Psikhiatr 2008, randomised 62 patients with GAD and neurasthenia to selank (n=30) versus the benzodiazepine medazepam (n=32). The abstract does not state the Selank dose or route, so those cells are n.a. here.

No human half-life, no injection-site data and no Western pharmacokinetic study were found in the sources fetched for this page. Reported evidence is real but thin and almost entirely Russian-language; treat published doses as trial documentation rather than a protocol.

04 / References

References

  1. Syunyakov T et al. Rapid and Slow Response During Treatment of GAD With Peptide Anxiolytic Selank. Eur Psychiatry 2012 ↗
  2. Zozulia AA et al. Efficacy and possible mechanisms of action of a new peptide anxiolytic selank in GAD and neurasthenia. 2008 (PubMed 18454096) ↗